Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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136
Tocris Bioscience™ MRT 68921 dihydrochloride
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ULK inhibitor
| Chemical Name or Material | N-[3-[[5-Cyclopropyl-2-[(1,2,3,4-tetrahydro-2-methyl-6-isoquinolinyl)amino]-4-pyrimidinyl]amino]propyl]cyclobutanecarboxamide dihydrochloride |
|---|---|
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C25H34N6O.2HCl |
| Formula Weight | Observed MW: 507.5 |
| Assay Percent Range | >98% |
137
Tocris Bioscience™ Phalloidin-FITC
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Green fluorescent cytoskeleton stain
138
Tocris Bioscience™ A 425619
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Potent TRPV1 antagonist
| Target | TRPV Antagonists |
|---|---|
| CAS | 581809-67-8 |
| Purity | >98% |
| Chemical Name or Material | N-5-Isoquinolinyl-N′-[[(4-(trifluoromethyl)phenyl]methyl]urea |
| Recommended Storage | Store at Room Temperature |
| Molecular Formula | C18H14F3N3O |
| Formula Weight | 345.32 |
139
Tocris Bioscience™ Bz 423
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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ATP synthase inhibitor; proapoptotic
| CAS | 216691-95-1 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Color | White |
| Solubility | Soluble to 100mM in DMSO and to 100mM in ethanol |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | 7-Chloro-1,3-dihydro-5-(4-hydroxyphenyl)-1-methyl-3-(2-naphthalenylmethyl)-2H-1,4-benzodiazepin-2-one |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C27H21ClN2O2 |
| Formula Weight | 440.92 |
140
Tocris Bioscience™ A37
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CAS: 896795-60-1 Molecular Formula: C21H25N3O3S2
| CAS | 896795-60-1 |
|---|---|
| Molecular Formula | C21H25N3O3S2 |
141
Tocris Bioscience™ ML 339
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Potent and selective hCXCR6 antagonist
| Target | Chemokine Receptor Antagonists |
|---|---|
| CAS | 2080300-49-6 |
| Product Type | Bioactive Small Molecule |
| Color | White |
| Solubility | Soluble to 100mM in DMSO and to 20mM in ethanol |
| Purity | 98% |
| Physical Form | Solid |
| Chemical Name or Material | N-[(1 R,3 S,5 S)-9-(2-((2-Chlorophenyl)amino)-2-exoethyl)-9-azabicyclo[3.3.1 ]nonan-3-yl)-3,4,5-trimethoxybenzamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C26H32ClN3O5 |
| Formula Weight | 502 |
142
Tocris Bioscience™ 3',3'-cGAMP sodium salt
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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STING agonist
143
Tocris Bioscience™ DMNPE-4 AM-caged-calcium
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Caged calcium
144
Tocris Bioscience™ BMS 986187, >98%
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 684238-37-7 Molecular Formula: C31H34O4
| CAS | 684238-37-7 |
|---|---|
| Molecular Formula | C31H34O4 |
145
Tocris Bioscience™ R 7050
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Inhibitor of TNF-α receptor 1 signaling
| Inhibitors | R 7050 |
|---|---|
| Product Type | R 7050 |
| Molecular Weight (g/mol) | 380.77 |
| Purity | >98% |
146
Tocris Bioscience™ AMG PERK 44
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Potent and selective PERK inhibitor; orally bioavailable
| Target | PERK Inhibitors |
|---|---|
| CAS | 1883548-84-2 |
| Purity | >98% |
| Chemical Name or Material | 4-[2-Amino-4-methyl-3-(2-methyl-6-quinolinyl)benzoyl]-1,2-dihydro-1-methyl-2,5-diphenyl-3H-pyrazol-3-one hydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C34H28N4O2.HCl |
| Formula Weight | 561.07 |
147
Tocris Bioscience™ LCB 03-0110 dihydrochloride
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Potent c-SRC kinase inhibitor; also inhibits DDR2, BTK and Syk
| Target | Src Family Kinase Inhibitors |
|---|---|
| Purity | >98% |
| Chemical Name or Material | 3-[[2-[3-(4-Morpholinylmethyl)phenyl]thieno[3,2-b]pyridin-7-yl]amino]phenol dihydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C24H23N3O2S.2HCl |
| Formula Weight | 490.45 |
148
Tocris Bioscience™ AZD 1480
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective JAK2 inhibitor; antiangiogenic
149
Tocris Bioscience™ GS 143
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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β-TrCP1 ligase inhibitor
| Target | Ubiquitin Ligase (E3) Inhibitors |
|---|---|
| CAS | 916232-21-8 |
| Purity | >98% |
| Chemical Name or Material | 4-[4-[[5-(2-Fluorophenyl)-2-furanyl]methylene]-4,5-dihydro-5-oxo-3-(phenylmethyl)-1H-pyrazol-1-yl]benzoic acid |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C28H19FN2O4 |
| Formula Weight | 466.46 |
150
Tocris Bioscience™ EML 425
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Reversible and non-competitive CBP/p300 inhibitor
| Target | Histone Acetyltransferase Inhibitors |
|---|---|
| CAS | 1675821-32-5 |
| Purity | >98% |
| Chemical Name or Material | 5-[(4-Hydroxy-2,6-dimethylphenyl)methylene]-1,3-bis(phenylmethyl)-2,4,6(1H,3H,5H)-pyrimidinetrione |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C27H24N2O4 |
| Formula Weight | 440.49 |