Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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136
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60,533
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136
R&D Systems™ DCLK1-IN-1
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable
137
R&D Systems™ Dooku 1
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Reversibly blocks Yoda1 activity; does not affect constitutive Piezo1 activity
| Target | Other Piezo Channel Compounds |
|---|---|
| CAS | 2253744-54-4 |
| Purity | 98% |
| Chemical Name or Material | 2-[(2,6-Dichlorobenzyl)thio)-5-(1 H-pyrrol-2-yl)-1,3,4-oxadiazole |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C13H9Cl2N3OS |
| Formula Weight | 326.2 |
138
R&D Systems™ KYP 2047
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. High affinity prolyl oligopeptidase inhibitor (Ki = 0.023 nM); anti-angiogenic, neuroprotective and brain penetrant
| CAS | 796874-99-2 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | (2S)-1-[[(2S)-1-(1-Oxo-4-phenylbutyl)-2-pyrrolidinyl]carbonyl]-2-pyrrolidinecarbonitrile |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C20H25N3O2 |
| Formula Weight | 339.44 |
139
R&D Systems™ BTD
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Selective TRPC5 activator
| CAS | 896684-04-1 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 6-Methyl-N-[3-(tricyclo[3.3.1.13,7]dec-1-yloxy)propyl]-4H-1,2,4-benzothiadiazine-3-propanamide-1,1-dioxide |
| Molecular Formula | C24H33N3O4S |
140
![R&D Systems™ Cy5-Fuc Labeled S2[3]f (Cy5-S2[3]f)](https://assets.fishersci.com/TFS-Assets/CCG/product-images/default.jpg-250.jpg)
R&D Systems™ Cy5-Fuc Labeled S2[3]f (Cy5-S2[3]f)
Used as a ligand for lectins and to study glycan protein interaction
141
R&D Systems™ ML T7
A Tocris product, part of R&D Systems. Inhibitor of phosphatidylserine/CEACAM1 binding to Tim-3
| Target | CEACAM1/CD66a |
|---|---|
| CAS | 459789-75-4 |
| Purity | 0.98 |
| Chemical Name or Material | 5-(2,4-Dichlorophenyl)-3a,6a-dihydro-3-(4-methylphenyl)spiro[1H-furo[3,4-c]pyrrole-1,2'-[2H]indene]-1',3',4,6(3H,5H)-tetrone |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C27H17Cl2NO5 |
142
R&D Systems™ ARCC 4 negative control
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Negative control for ARCC 4 (Cat. No. 7254)
143
R&D Systems™ EM 12-FS
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Molecular glue; induces degradation of NQAT1
| Target | Molecular Glues |
|---|---|
| CAS | 2839138-44-0 |
| Purity | 0.95 |
| Chemical Name or Material | 3-[6-[(Fluorosulfonyl)oxy]-1,3-dihydro-1-oxo-2H-isoindol-2-yl]-2,6-piperidinedione |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C13H11FN2O6S |
144
R&D Systems™ Pomalidomide 4'-alkylC6-azide
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Cereblon ligand with alkyl linker and terminal azide for onward chemistry
145
| CAS | 7770-78-7 |
|---|---|
| Molecular Formula | C21H24O6 |
146
R&D Systems™ Silodosin
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Selective α1A adrenoceptor antagonist (Ki = 0.036 nM)
| CAS | 160970-54-7 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 2,3-Dihydro-1-(3-hydroxypropyl)-5-[(2R)-2-[[2-[2-(2,2,2-trifluoroethoxy)phenoxy]ethyl]amino]propyl]-1H-indole-7-carboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H32F3N3O4 |
| Formula Weight | 495.53 |
147
R&D Systems™ Dapansutrile
A Tocris product, part of R&D Systems. NLRP3 inflammasome inhibitor; disrupts inflammasome formation
| Product Type | Inhibitor |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C4H7NO2S |
| Formula Weight | 133.17 |
148
R&D Systems™ AF 64394
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective GPR3 inverse agonist
| CAS | 1637300-25-4 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[[4-Chloro-2-(1-methylethoxy)phenyl]methyl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
| Molecular Formula | C21H20ClN5O |
