Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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136
Tocris Bioscience™ UoS 12258
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Positive allosteric modulator of AMPA receptors (pEC50 = 5.2 for potentiation of AMPA-mediated currents in vitro)
| CAS | 875927-64-3 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[(2S)-5-(6-Fluoro-3-pyridinyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C17H19FN2O2S |
| Formula Weight | 334.41 |
139
Tocris Bioscience™ Ivabradine hydrochloride
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Greener Choice
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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HCN channel blocker; inhibits If pacemaker current
| CAS | 148849-67-6 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 3-[3-[[[(7S)-3,4-Dimethoxybicyclo[4.2.0]octa-1,3,5-trien-7-yl]methyl]methylamino]propyl]-1,3,4,5-tetrahydro-7,8-dimethoxy-2H-3-benzazepin-2-one hydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C27H36N2O5.HCl |
140
Tocris Bioscience™ SAK 3
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent CaV3.1/3.3 activator; orally bioavailable
| Target | Cav3.x Channel Activators |
|---|---|
| CAS | 1256269-87-0 |
| Purity | 98% |
| Chemical Name or Material | Ethyl 8′-methyl-2′,4-dioxo-2-(piperidin-1-yl)-2′H-spiro[cyclopent[2]ene-1,3′-imidazo[1,2-a]pyridine]-3-carboxylate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C20H23N3O4 |
141
Tocris Bioscience™ Pomalidomide 4'-alkylC6-azide
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Cereblon ligand with alkyl linker and terminal azide for onward chemistry
142
| CAS | 7770-78-7 |
|---|---|
| Molecular Formula | C21H24O6 |
143
Tocris Bioscience™ Darapladib
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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Potent lp-PLA2 inhibitor
| CAS | 356057-34-6 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[2-(Diethylamino)ethyl]-2-[[(4-fluorophenyl)methyl]thio]-4,5,6,7-tetrahydro-4-oxo-N-[[4'-(trifluoromethyl)[1,1'-biphenyl]-4-yl]methyl]-1H-cyclopentapyrimidine-1-acetamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C36H38F4N4O2S |
| Formula Weight | 666.77 |
144
| CAS | 84-26-4 |
|---|---|
| Molecular Formula | C18H13N3O |
145
Tocris Bioscience™ CRBN PROTAC™ 14a
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Cereblon Degrader (PROTAC™)
146
Tocris Bioscience™ PZM21
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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Small and/or specialty supplier based on Federal laws and SBA requirements.
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Selective μ receptor agonist
| Target | mu Opioid Receptor Agonists |
|---|---|
| CAS | 1997387-43-5 |
| Purity | 0.98 |
| Chemical Name or Material | N-[(2 S)-2-(Dimethylamino)-3-(4-hydroxyphenyl)propyl]-N'-[(1 S)-1-methyl-2-(3-thienyl)ethyl]urea |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H27N3O2S |
147
Tocris Bioscience™ tri-GalNAc COOH
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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Asialoglycoprotein receptor ligand with PEG linker and carboxylic acid group for onward chemistry
148
Tocris Bioscience™ Cholesterol
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Component of lipid nanoparticles (LNPs); modulator of lipid bilayer fluidity
149
Tocris Bioscience™ AZ 12799734
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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Small and/or specialty supplier based on Federal laws and SBA requirements.
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Potent TGF-βRI inhibitor
| CAS | 1117684-36-2 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 4-[[4-[(2.6-Dimethyl-3-pyridinyl)oxy]-2-pyridinyl]amino]benzenesulfonamide |
| Molecular Formula | C18H18N4O3S |
150
Tocris Bioscience™ Tazemetostat
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Potent and selective EZH2 inhibitor
| Target | EZH2 Inhibitor |
|---|---|
| CAS | 1403254-99-8 |
| Purity | 0.97 |
| Chemical Name or Material | N-[(1,2-Dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-5-[ethyl(tetrahydro-2H-pyran-4-yl)amino]-4-methyl-4'-(4-morpholinylmethyl)[1,1'-biphenyl]-3-carboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C34H44N4O4 |